Enzymology in drug discovery [electronic resource] : part 2 of 2 / Robert A. Copeland.
Material type:
FilmSeries: Henry Stewart talksBiomedical & life sciences collection. Small molecule drug discovery: Publisher: London : Henry Stewart Talks, 2013Description: 1 online resource (1 streaming video file (66 min.) : color, sound)Other title: Enzymology in drug discovery part, part 2 of 2Subject(s): Drugs -- Design | Enzyme inhibitors -- Structure-activity relationships | Enzyme inhibitors -- Therapeutic use | Enzymes | Enzymology | Pharmaceutical chemistry | Drug Design | Drug Discovery | Enzyme Inhibitors -- chemistry | Enzyme Inhibitors -- metabolism | Enzyme Inhibitors -- pharmacology | Enzyme Inhibitors -- therapeutic useOnline resources: Click here to access online | Series Animated audio-visual presentation with synchronized narration.
Title from title frames.
Contents: Enzymes as targets for drug discovery -- Protein-ligand binding equilibria -- Enzyme reaction mechanisms -- Structure and function of enzyme active sites -- Measuring enzyme velocity in the laboratory -- Reversible modes of enzyme inhibition -- Enzyme inhibition as a mechanism of pharmacological intervention in disease -- Clinical value of different inhibition modalities -- Non-classical inhibition -- Enzyme assays and screening criteria -- Lead optimization -- Summary: basic information to look for.
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Mode of access: World Wide Web.