Sim, Edith,

Arylamine N-acetyltransferases part 3 of 3 / [electronic resource] : Arylamine N-acetyltransferases 3 Edith Sim. - London : Henry Stewart Talks, 2016. - 1 online resource (1 streaming video file (19 min.) : color, sound). - Drug metabolizing enzymes : fundamentals, study methods, recent advances and clinical significance, 2056-452X . - Henry Stewart talks. Biomedical & life sciences collection. Drug metabolizing enzymes : fundamentals, study methods, recent advances and clinical significance. .

Animated audio-visual presentation with synchronized narration. Title from title frames. Updated version of a talk first published in 2007.

Contents: Mechanism of action -- Reaction substrates -- Isoform substrate profiles -- Isoenzymes NAT1 and NAT2 -- Regulation of gene expression -- Pharmacogenetics -- Phenotype/genotype correlation -- Ethnic variation -- Transgenic mouse models -- NAT protein structures -- NAT as a biomarker in breast cancer -- NAT inhibitors as diagnostic agents -- NAT in mycobacteria -- NAT inhibitors as an approach to potential anti-tubercular agents.

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Mode of access: World Wide Web.

4279 Henry Stewart Talks


Antibacterial agents.
Biochemical markers.
Breast--Cancer.
Drug development.
Drugs--Metabolism.
Enzyme Inhibitors.
Isoenzymes.
Transferases.
Antitubercular Agents.
Arylamine N-Acetyltransferase--antagonists & inhibitors.
Arylamine N-Acetyltransferase--genetics.
Arylamine N-Acetyltransferase--metabolism.
Bacterial Infections--drug therapy.
Biomarkers.
Breast Neoplasms--diagnosis.
Drug Discovery--methods.
Enzyme Inhibitors--pharmacology.
Ethnic Groups.
Gene Expression Regulation, Enzymologic.
Genetic Association Studies.
Isoenzymes--metabolism.
Mice, Transgenic.
Mycobacterium--drug effects.
Pharmaceutical Preparations--metabolism.
Pharmacogenetics.
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